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Pharmacokinetic and Permeation Studies in Rat Brain of Natural Compounds Led to Investigate Eugenol as Direct Activator of Dopamine Release in PC12 Cells
Pavan, Barbara; Bianchi, Anna; Botti, Giada; Ferraro, Luca; Valerii, Maria Chiara; Spisni, Enzo; Dalpiaz, Alessandro     dettagli >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 24, No. 2, pp: 1800-1-1800-24, Anno: 2023

Improving in vivo oral bioavailability of a poorly soluble drug: a case study on polymeric versus lipid nanoparticles
Rassu, Giovanna; Obinu, Antonella; Serri, Carla; Piras, Sandra; Carta, Antonio; Ferraro, Luca; Gavini, Elisabetta; Giunchedi, Paolo; Dalpiaz, Alessandro     dettagli >>
DRUG DELIVERY AND TRANSLATIONAL RESEARCH
Vol. 13, No. 4, pp: 1128-1139, Anno: 2023

Delivering hydrosoluble compounds through the skin: what are the chances?
Demartis, S; Rassu, G; Mazzarello, V; Larrañeta, E; Hutton, A; Donnelly, R F; Dalpiaz, A; Roldo, M; Guillot, A J; Melero, A; Giunchedi, P; Gavini, E     dettagli >>
INTERNATIONAL JOURNAL OF PHARMACEUTICS
Vol. 646, No. 1, pp: 123457-1-123457-18, Anno: 2023

Dimeric ferulic acid conjugate as a prodrug for brain targeting after nasal administration of loaded solid lipid microparticles
Botti, Giada; Bianchi, Anna; Dalpiaz, Alessandro; Tedeschi, Paola; Albanese, Valentina; Sorrenti, Milena; Catenacci, Laura; Bonferoni, Maria Cristina; Beggiato, Sarah; Pavan, Barbara     dettagli >>
EXPERT OPINION ON DRUG DELIVERY
Vol. 20, No. 1, pp: 1657-1679, Anno: 2023

Conjugation, Prodrug, and Co-Administration Strategies in Support of Nanotechnologies to Improve the Therapeutic Efficacy of Phytochemicals in the Central Nervous System
Rassu, Giovanna; Sorrenti, Milena; Catenacci, Laura; Pavan, Barbara; Ferraro, Luca; Gavini, Elisabetta; Cristina Bonferoni, Maria; Giunchedi, Paolo; Dalpiaz, Alessandro     dettagli >>
PHARMACEUTICS
Vol. 15, No. 6, pp: 1578-1-1578-43, Anno: 2023

Effects of Microencapsulated Ferulic Acid or Its Prodrug Methyl Ferulate on Neuroinflammation Induced by Muramyl Dipeptide
Botti, Giada; Bianchi, Anna; Pavan, Barbara; Tedeschi, Paola; Albanese, Valentina; Ferraro, Luca; Spizzo, Federico; Del Bianco, Lucia; Dalpiaz, Alessandro     dettagli >>
INTERNATIONAL JOURNAL OF ENVIRONMENTAL RESEARCH AND PUBLIC HEALTH
Vol. 19, No. 17, pp: 10609-1-10609-24, Anno: 2022

Cocrystals of Nitrofurantoin: How Coformers Can Modify Its Solubility and Permeability Across Intestinal Cell Monolayers
Segalina, A.; Pavan, B.; Ferretti, V.; Spizzo, F.; Botti, G.; Bianchi, A.; Pastore, M.; Dalpiaz, A.     dettagli >>
CRYSTAL GROWTH & DESIGN
Vol. 22, No. 5, pp: 3090-3106, Anno: 2022

Nasal biocompatible powder of Geraniol oil complexed with cyclodextrins for neurodegenerative diseases: physicochemical characterization and in vivo evidences of nose to brain delivery
Truzzi, E.; Rustichelli, C.; de Oliveira Junior, E. R.; Ferraro, L.; Maretti, E.; Graziani, D.; Botti, G.; Beggiato, S.; Iannuccelli, V.; Lima, E. M.; Dalpiaz, A.; Leo, E.     dettagli >>
JOURNAL OF CONTROLLED RELEASE
Vol. 335, No. 1, pp: 191-202, Anno: 2021

Chitosan/heparin polyelectrolyte complexes as ion-paring approach to encapsulate heparin in orally administrable SLN: In vitro evaluation
Maretti, E.; Pavan, B.; Rustichelli, C.; Montanari, M.; Dalpiaz, A.; Iannuccelli, V.; Leo, E.     dettagli >>
COLLOIDS AND SURFACES. A, PHYSICOCHEMICAL AND ENGINEERING ASPECTS
Vol. 608, No. 1, pp: 125606-1-125606-11, Anno: 2021

Targeting systems to the brain obtained by merging prodrugs, nanoparticles, and nasal administration
Botti, G.; Dalpiaz, A.; Pavan, B.     dettagli >>
PHARMACEUTICS
Vol. 13, No. 8, pp: 1144-1-1144-31, Anno: 2021

Polymeric nanomicelles based on inulin D α-tocopherol succinate for the treatment of diabetic retinopathy
Rassu, G.; Pavan, B.; Mandracchia, D.; Tripodo, G.; Botti, G.; Dalpiaz, A.; Gavini, E.; Giunchedi, P.     dettagli >>
JOURNAL OF DRUG DELIVERY SCIENCE AND TECHNOLOGY
Vol. 61, No. 1, pp: 102286-1-102286-10, Anno: 2021

Versatile nasal application of cyclodextrins: Excipients and/or actives?
Rassu, G.; Sorrenti, M.; Catenacci, L.; Pavan, B.; Ferraro, L.; Gavini, E.; Bonferoni, M. C.; Giunchedi, P.; Dalpiaz, A.     dettagli >>
PHARMACEUTICS
Vol. 13, No. 8, pp: 1180-1-1180-23, Anno: 2021

Effect of a fiber d-limonene-enriched food supplement on intestinal microbiota and metabolic parameters of mice on a high-fat diet
Valerii, M. C.; Turroni, S.; Ferreri, C.; Zaro, M.; Sansone, A.; Dalpiaz, A.; Botti, G.; Ferraro, L.; Spigarelli, R.; Bellocchio, I.; D'Amico, F.; Spisni, E.     dettagli >>
PHARMACEUTICS
Vol. 13, No. 11, pp: 1753-1-1753-17, Anno: 2021

Cancer stem cells and nanomedicine: new opportunities to combat multidrug resistance?
Dalpiaz, A.; Paganetto, G.; Botti, G.; Pavan, B.     dettagli >>
DRUG DISCOVERY TODAY
Vol. 25, No. 9, pp: 1651-1667, Anno: 2020

Design and formulation of Eudragit-coated zein/pectin nanoparticles for the colon delivery of resveratrol
Contado, C.; Caselotto, L.; Mello, P.; Maietti, A.; Marvelli, L.; Marchetti, N.; Dalpiaz, A.     dettagli >>
EUROPEAN FOOD RESEARCH AND TECHNOLOGY
Vol. 246, No. 12, pp: 2427-2441, Anno: 2020

Solid lipid nanoparticles as formulative strategy to increase oral permeation of a molecule active in multidrug-resistant tuberculosis management
Obinu, A.; Porcu, E. P.; Piras, S.; Ibba, R.; Carta, A.; Molicotti, P.; Migheli, R.; Dalpiaz, A.; Ferraro, L.; Rassu, G.; Gavini, E.; Giunchedi, P.     dettagli >>
PHARMACEUTICS
Vol. 12, No. 12, pp: 1132-1-1132-24, Anno: 2020

Nasal administration of nanoencapsulated geraniol/ursodeoxycholic acid conjugate: Towards a new approach for the management of Parkinson's disease
de Oliveira Junior, E. R.; Truzzi, E.; Ferraro, L.; Fogagnolo, M.; Pavan, B.; Beggiato, S.; Rustichelli, C.; Maretti, E.; Lima, E. M.; Leo, E.; Dalpiaz, A.     dettagli >>
JOURNAL OF CONTROLLED RELEASE
Vol. 321, No. 10 May 2020, pp: 540-552, Anno: 2020

Exploring the use of spray congealing to produce solid dispersions with enhanced indomethacin bioavailability: In vitro characterization and in vivo study
Bertoni, Serena; Albertini, Beatrice; Ferraro, Luca; Beggiato, Sarah; Dalpiaz, Alessandro; Passerini, Nadia     dettagli >>
EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
Vol. 139, No. 1, pp: 132-141, Anno: 2019

Bile salt-coating modulates the macrophage uptake of nanocores constituted by a zidovudine prodrug and enhances its nose-to-brain delivery
Dalpiaz, A.; Fogagnolo, M.; Ferraro, L.; Beggiato, S.; Hanuskova, M.; Maretti, E.; Sacchetti, F.; Leo, E.; Pavan, B.     dettagli >>
EUROPEAN JOURNAL OF PHARMACEUTICS AND BIOPHARMACEUTICS
Vol. 144, No. 1, pp: 91-100, Anno: 2019

Drug release from pharmaceutical co-crystals: Are therapeutic and safety properties of active pharmaceutical substances retained?
Dalpiaz, A.; Ferretti, V.; Botti, G.; Pavan, B.     dettagli >>
CURRENT DRUG DELIVERY
Vol. 16, No. 6, pp: 486-489, Anno: 2019

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